Journal of Medicinal Chemistry
Volume 42, Issue 3 (February 11, 1999)
Copyright © 1999
American Chemical Society
| COMMUNICATIONS TO THE EDITOR | |
333-335 | A New Single-Photon Emission Computed Tomography Imaging Agent for Serotonin Transporters: [123I]IDAM, 5-Iodo-2-((2-((dimethylamino)methyl)phenyl)thio)benzyl Alcohol
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ARTICLES | |
336-345 | Effect of Modifications of the Alkylpiperazine Moiety of Trazodone on 5HT2A and  1 Receptor Binding Affinity
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346-355 | N-Substituted 2-(2,6-Dinitrophenylamino)propanamides: Novel Prodrugs That Release a Primary Amine via Nitroreduction and Intramolecular Cyclization
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356-363 | Identification and Characterization of m1 Selective Muscarinic Receptor Antagonists
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364-372 | Ajoene Is an Inhibitor and Subversive Substrate of Human Glutathione Reductase and Trypanosoma cruzi Trypanothione Reductase: Crystallographic, Kinetic, and Spectroscopic Studies
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373-380 | Three-Dimensional Quantitative Structure-Activity Relationship of Interleukin 1- Converting Enzyme Inhibitors: A Comparative Molecular Field Analysis Study
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381-392 | Antitumor Benzothiazoles. 7. Synthesis of 2-(4-Acylaminophenyl)benzothiazoles and Investigations into the Role of Acetylation in the Antitumor Activities of the Parent Amines
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393-399 | The Presence of Substituents on the Aryl Moiety of the Aryl Phosphoramidate Derivative of d4T Enhances Anti-HIV Efficacy in Cell Culture: A Structure-Activity Relationship
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400-404 | Dermorphin and Deltorphin Glycosylated Analogues: Synthesis and Antinociceptive Activity after Systemic Administration
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405-408 | Design of Antineoplastic Agents Based on the "2-Phenylnaphthalene-Type" Structural Pattern. 4. Synthesis and Biological Activity of 2-Chloro-3-(substituted phenoxy)-1,4-naphthoquinones and Related 5,8-Dihydroxy-1,4-naphthoquinones
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409-414 | A New Class of Pseudopeptide Antagonists of the Kinin B1 Receptor Containing Alkyl Spacers
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415-426 | Structure-Activity Studies of Conantokins as Human N-Methyl-D-aspartate Receptor Modulators
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427-437 | Synthesis, Pharmacological Evaluation, and Structure-Activity Relationship and Quantitative Structure-Activity Relationship Studies on Novel Derivatives of 2,4-Diamino-6,7-dimethoxyquinazoline 1-Adrenoceptor Antagonists
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438-445 | Allosteric Interactions of Quaternary Strychnine and Brucine Derivatives with Muscarinic Acetylcholine Receptors
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446-457 | Synthesis of Cytotoxic Indenoisoquinoline Topoisomerase I Poisons
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458-477 | Three-Dimensional Quantitative Structure-Activity Relationship Analyses Using Comparative Molecular Field Analysis and Comparative Molecular Similarity Indices Analysis To Elucidate Selectivity Differences of Inhibitors Binding to Trypsin, Thrombin, and Factor Xa
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478-489 | Flavonoid-Related Modulators of Multidrug Resistance: Synthesis, Pharmacological Activity, and Structure-Activity Relationships
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490-496 | 1-Aryl-4-[(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and Their Analogues: Influence of the Stereochemistry of the Tetrahydronaphthalen-1-yl Nucleus on 5-HT1A Receptor Affinity and Selectivity versus 1 and D2 Receptors. 5
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497-509 | Structure-Activity Relationships: Analogues of the Dicaffeoylquinic and Dicaffeoyltartaric Acids as Potent Inhibitors of Human Immunodeficiency Virus Type 1 Integrase and Replication
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510-514 | Novel Antitumor 2-Cyanoaziridine-1-carboxamides
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515-525 | Metallopeptidase Inhibitors of Tetanus Toxin: A Combinatorial Approach
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BRIEF ARTICLES | |
526-531 | N-Methyl-5-tert-butyltryptamine: A Novel, Highly Potent 5-HT1D Receptor Agonist
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BOOK REVIEWS | |
532-532 | How To Find Chemical Information: A Guide for Practicing Chemists, Educators, and Students, 3rd Edition By Robert E. Maizell. John Wiley & Sons, Inc., New York. 1998. xxiii + 515 pp. 16 × 23 cm. ISBN 0-471-125792. $64.95.
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